Representative nuclei stained by eu are shown 22 h after 2 h treatment with 25 µg ml cisplatin. Compound 401是dna pk和mtor抑制剂 ic50分别为0 28 μm和5 3 μm 它对p110α p85α pi3k没有明显抑制作用 在cos7细胞中抑制s6激酶在thr389位的磷酸化和akt在ser473位的磷酸化 s3901.
dna pk activity sensitizes a549 cells
nature
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